Home   >  
Protease/Metabolic Enzyme
  >  
Pyruvate Kinase
  >   PKM2 inhibitor
PKM2 inhibitor Chemical Structure

PKM2 inhibitor

Data Sheet For research use only. Not for human use.
Cat. No. :BCP23555CAS No. :94164-88-2Purity:98%
 Tel: 0086-17754423994   or   orders@biochempartner.com
Real-Time Inquiry ×

* Required Fields.

Please complete the form below and you will get the price list in 1 minute.

Product name

 

* Applicant name

Catalog Number

 

* Institution/Company

* Email address

 

Phone number

Country

 

* Quantity Required

Remarks

Inquiry Online ×

* Required Fields.

Please complete the form below and we will contact you shortly.

Product name

 

* Applicant name

Catalog Number

 

* Institution/Company

* Email address

 

Phone number

Country

 

* Quantity Required

Remarks

Bulk Inquiry ×

* Required Fields.

Please complete the form below and we will contact you shortly.

Product name

 

* Applicant name

Catalog Number

 

* Institution/Company

* Email address

 

Phone number

Country

 

* Quantity Required

Remarks

  • Chemical Properties&Biological Activity
CAS No. 94164-88-2 Cat. No. BCP23555
Name PKM2 inhibitor
Synonyms MDK4882; MDK-4882; MD K4882;PKM2-IN-1;
SMILES
Chemical Name
Formula C18H19NO2S2 M. Wt 345.48
Purity 98% Storage Store at 4-8°C
Description PKM2 inhibitor also known as MDK4882 or PKM2-IN-1 , is a PKM2 inhibitor. MDK4882 was first described in Eur J Med Chem. 2017;138:343-352. Currently there is no formal name. We temporally name it as MDK4882 for the convenience of communication, in which the last 4 digit of CAS# is used. MDK4882 displayed potent PKM2 inhibitory activity than the reported optimal PKM2 inhibitor shikonin. MDK4882 also showed nanomolar antiproliferative activity toward a series of cancer cell lines with high expression of PKM2 including HCT116, Hela and H1299 with IC50 values ranging from 0.18 to 1.56 μM. MDK4882 exhibited more cytotoxicity on cancer cells than normal cells.
  • Quality Control&Technical Support
In the process of purchasing and using Biochempartner products, you can consult us if you have any problems: orders@biochempartner.com. We will try our best to solve all your doubts.

Recommend Products

More >

Tags:PKM2 inhibitor supplier,PKM2 inhibitor purchase,PKM2 inhibitor manufacturer,PKM2 inhibitor distributor,PKM2 inhibitor cost,PKM2 inhibitor buy,PKM2 inhibitor for sale

0086-13720134139