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Nature products
Antibodies
Peptides
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Intermediate
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Raw Materials
Epigenetic Reader Domain
Chemical Structure | Cat. No. | Product Name | CAS No. |
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BCP23818 | PFI-4 New | 900305-37-5 | |
PFI-4 is a potent and highly selective BRPF1 Bromodomain (BRPF1B) inhibitor, with an IC50 of 172 nM. PFI-4 can be used to explore the functional mechanisms of the HBO1/BRPF1 complex and to study bone loss and osteolytic malignant bone lesions.
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BCP23999 | BAZ2-ICR New | 1665195-94-7 | |
BAZ2-ICR is a potent, selective, cell active and orally active BAZ2A/B bromodomains inhibitor with IC50s of 130 nM and 180 nM, and Kds of 109 nM and 170 nM, respectively. BAZ2-ICR shows 10-15-fold selectivity for binding BAZ2A/B over CECR2 and >100-fold selectivity over all other bromodomains. BAZ2-ICR is an epigenetic chemical probe.
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BCP25147 | BMS 986158 New | 1800340-40-2 | |
BMS-986158 is an inhibitor of the bromodomain and extra-terminal (BET) proteins.
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BCP48567 | SRX3177 New | 2241237-51-2 | |
SRX3177 is a novel potent triple action inhibitor, targeting BRD, PI3K, and CDK.
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BCP46987 | AU-15330 New | 2380274-50-8 | |
AU-15330 is a novel, highly specific and VHL-dependent PROTAC degrader of SWI/SNF ATPase components (SMARCA2, SMARCA4 and PBRM1) that shows preferential cytotoxicity in enhancer-binding transcription factor-addicted cancers at low nanomolar concentrations.
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BCP46797 | EML 425 New | 1675821-32-5 | |
EML425 is a potent and selective CREB binding protein (CBP)/p300 inhibitor with IC50s of 2.9 and 1.1 μM, respectively.
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BCP46564 | CFT-8634 New | 2704617-96-7 | |
CFT-8634 is a degrader targeting BRD9 extracted from patent WO2021178920A1 compound 173.
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BCP46513 | GSK1379725A New | 1802251-00-8 | |
GSK1379725A is the first selective inhibitor of BPTF over Brd4.
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BCP46449 | BAZ1A-IN-1 New | 941521-45-5 | |
BAZ1A-IN-1 is a potent inhibitor of BAZ1A (bromodomain-containing protein). BAZ1A-IN-1 shows a KD value of 0.52 μM against BAZ1A bromodomain.
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BCP46311 | M-525 New | 2173582-08-4 | |
M-525 is a first-in-class, highly potent, irreversible small-molecule inhibitor of the menin-MLL interaction.
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