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CAS号 | 1137916-97-2 | 货号 | BCP25241 |
关联产品 | 752240-01-0(MK-0941) | ||
中文名 | MK-0941 mesylate | ||
英文名 | MK-0941 mesylate | ||
中文别名 | |||
英文别名 | MK-0941; MK 0941 mesylate; MK0941 mesylate; | ||
SMILES | O=C(NC1=NN(C)C=C1)C2=CC(O[C@@H](C)CO)=CC(OC3=CC=C(S(=O)(CC)=O)N=C3)=C2.OS(=O)(C)=O | ||
化学名称 | |||
分子式 | C21H24N4O6S.CH4O3S | 分子量 | 556.61 |
纯度 | 98% | 配送 | 惯例下常温包邮 |
产品描述 | MK-0941 mesylate (MK0941) is a novel potent, orally active Glucokinase (GK) activator with EC50 of 0.240 and 0.065 uM in 2.5 and 10 mM glucose, respectively; increases insulin secretion by 17-fold and glucose uptake up to 18-fold, respectively, in isolated rat islets of Langerhans and hepatocytes at 10 uM; exhibits strong glucose-lowering activity in rodent models of type 2 diabetes and healthy dogs. |
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