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Estrogen Receptor

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Estrogen Receptor

结构式 货号 产品名称 CAS号
OP-1250 结构式
 BCP49307 OP-1250 OP-1250
OP-1250 is a novel oral compound developed to completely antagonize the estrogen receptor (ER) and block the ER-mediated cancer cell growth and proliferation signal.
Camizestrant 结构式
 BCP48205 Camizestrant 2222844-89-3
Camizestrant is an orally available selective estrogen receptor degrader (SERD), with potential antineoplastic activity. Upon administration, SERD AZD9833 binds to the estrogen receptor (ER) and induces a conformational change that results in the degradation of the receptor. This prevents ER-mediated signaling and inhibits the growth and survival of ER-expressing cancer cells.
Fispemifene 结构式
 BCP23860 Fispemifene 341524-89-8
Fispemifene is a selective estrogen receptor modulator (SERM) potentially for the treatment of hypogonadism.
Endoxifen hydrochloride 结构式
 BCP24689 因多昔芬盐酸盐 1197194-41-4
Endoxifen HCl, the active metabolite of Tamoxifen, ia a potent and selective estrogen receptor antagonist. Phase 2.
Methylpiperidino pyrazole 结构式
 BCP48025 Methylpiperidino pyrazole 289726-02-9
Methylpiperidino pyrazole is a high-affinity and selective ERα antagonist, exhibiting 200-fold potency for ERα over ERβ.
H3B-6545 Hydrochloride 结构式
 BCP48272 H3B-6545 Hydrochloride 2052132-51-9
H3B-6545 Hydrochloride is a selective, oral estrogen receptor covalent antagonist (SERCA).
2-Hydroxyestrone 结构式
 BCP46743 2-羟雌甾酮 362-06-1
2-Hydroxyestrone, a specific receptor-mediated antiestrogenic agent with anticarcinogenic activity, inhibits the proliferation of estrogen receptor-positive MCF-7, but not estrogen receptor-negative MDA-MB-231.
ARV-471 结构式
 BCP45881 ARV-471 2229711-08-2
ARV-471 is a best-in-class, orally active estrogen receptor (ER) PROTAC degrader.
Amcenestrant 结构式
 BCP38455 Amcenestrant 2114339-57-8
Amcenestrant (SAR439859) is an orally available and nonsteroidal selective estrogen receptor degrader (SERD) with potential antineoplastic activity. SAR439859 is a potent estrogen receptor (ER) antagonist with EC50 of 0.2 nM for ERα degradation.
Giredestrant tartrate 结构式
 BCP43932 Giredestrant tartrate 2407529-33-1
Giredestrant, also known as GDC-9545 and RG6171, is a SERD.
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