所有产品分类
所有产品
信号通路
- Angiogenesis/Protein Tyrosine Kinase
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GPCR/G Protein
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Neuro Signaling Pathway
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Protease/Metabolic Enzyme
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研究领域
- Metabolic Disease
- Neurological Disease
- Endocrinology
- Diabetes
- Cardiovascular Disease
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- Inflammation
- Infection
- Cancer
天然产物
抗体
多肽
催化剂
杂质对照品
医药中间体
基础原料
LXR
| 结构式 | 货号 | 产品名称 | CAS号 |
|---|
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BCP24282 | GSK9772 新 | 928035-84-1 |
GSK9772 is a novel potent transrepression-selective liver X receptor modulator with anti-inflammatory activity.
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BCP49028 | DMHCA 新 | 79066-03-8 |
DMHCA is a gene-selective LXR modulator that mediates potent transcriptional activation of ABCA1 gene expression.
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BCP39540 | GSK 2033 新 | 1221277-90-2 |
GSK2033 is a LXR antagonist with pIC50s of 7 and 7.4 for LXRα or LXRβ, respectively.
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BCP42686 | LXRβ agonist-2 新 | 1949801-52-8 |
LXRβ agonist-2 is a highly potent and β-selective liver X receptor (LXRβ) agonist with EC50 of 7 nM.
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BCP31854 | RGX-104 新 | 610318-54-2 |
RGX-104 is an orally bioavailable and potent liver-X nuclear hormone receptor (LXR) agonist that modulates innate immunity via transcriptional activation of the ApoE gene.
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BCP29451 | RGX-104 HCl | 610318-03-1 |
RGX-104 is a small-molecule LXR agonist that modulates innate immunity via transcriptional activation of the ApoE gene.
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BCP20751 | BMS-779788 | 918348-67-1 |
BMS-779788 is a LXR partial agonist with IC50 values of 68 nM for LXRα and 14 nM for LXRβ.
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BCP23542 | BMS-852927 | 1256918-39-4 |
BMS-852927 is an LXRβ-selective agonist.
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BCP19166 | AZ-876 | 898800-26-5 |
AZ876 is a novel high-affinity LXR agonist. AZ876 was 25-fold and 2.5-fold more potent than GW3965 (HY-10627) on human (h)LXRα and hLXRβ respectively.
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BCP15765 | SR-9243 | 1613028-81-1 |
SR9243 is a liver-X-receptor (LXR) inverse agonist that induces LXR-corepressor interaction.
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