CL 316243
CAS号 | 138908-40-4 | 货号 | BCP44544 |
中文名 | CL 316243 | ||
英文名 | CL 316243 | ||
中文别名 | |||
英文别名 | CL 316243; CL316243; CL-316,243; CL 316,243; CL316,243. HP 186; HP-186; HP186; | ||
分子式 | C20H18ClNO7.2Na | 分子量 | 465.79 |
生物活性 | CL-316243 is a potent and highly selective β3-adrenoceptor agonist (EC50 = 3 nM); > 10000-fold selective over β1 and β2 receptors. CL-316243 restores the expression of down-regulated fatty acid oxidation genes in type 2 diabetic mice. CL-316,243 enhances insulin-stimulated glucose disposal in nonobese rats. CL 316243 possesses anti-obesity and anti-diabetic effects and consequently may be useful for treating obesity as well as non-insulin-dependent diabetes mellitus in obese persons, without causing excessive side effects. | ||
信号通路 | Neuro Signaling Pathway GPCR/G Protein | ||
靶 点 | Adrenergic Receptor |
结构式
本页面部分数据来自于公开的网络资源,所以瀚香生物不能保证其准确性。
不同批次的产品详情请咨询我们的客服:
- 全国免费电话:400-099-8200
瀚香生物(Biochempartner) 的所有产品和服务仅用于科学研究,禁止用于人体和治疗!