RVX297

  • 化学数据
CAS号 1044871-04-6 货号 BCP43937
中文名 RVX297
英文名 RVX297
中文别名
英文别名 RVX 297; RVX-297;
分子式 C24H29N3O4 分子量 423.5
  • 用途
生物活性 RVX-297 is a BD2 selective inhibitor of BET bromodomains. RVX-297 is structurally related to the clinical compound RVX-208, currently undergoing phase III clinical trials for the treatment of cardiovascular diseases, but is distinctly different in its biological and pharmacokinetic profiles. RVX-297 preferentially binds to the BD2 domains of the BET bromodomain and Extra Terminal (BET) family of protein. Selective inhibition of either BD1 or BD2 can have significant implications on differential gene expression, which possibly can be further linked to the specific disease indication.
信号通路 Epigenetics 
靶 点 Epigenetic Reader Domain 

结构式

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